Product name : AM-251 (AM251, AM 251)
Product No. : CS-985
Price : 100mg, $675, 500mg/$1875
CAS :
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Details: |
AM251 (CAS: 183232-66-8) is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also potent GPR55 agonist (EC50 = 39 nM).
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